Published January 1, 2017 | Version v1
Journal article Open

Synthesis of Novel Benzothiazole-Piperazine Derivatives and Their Biological Evaluation as Acetylcholinesterase Inhibitors and Cytotoxic Agents

  • 1. Yeditepe Univ, Fac Pharm, Dept Pharmaceut Chem, TR-34755 Istanbul, Turkey
  • 2. Eastern Mediterranean Univ, Fac Pharm, Dept Pharmaceut Chem, Famagusta, Northern Cyprus, Turkey
  • 3. Middle East Tech Univ, Grad Sch Informat, Bioinformat Dept, Ankara, Turkey
  • 4. Martin Luther Univ Halle Wittenberg, Inst Pharm, Med Chem Dept, Halle, Saale, Germany

Description

Objective and Method: A new series of benzothiazole-piperazine derivatives was synthesized and a complete chemical characterization of the novel compounds was provided. In vitro cytotoxic activities were screened against colorectal (HCT-116), breast (MCF-7) and hepatocellular (Huh7) cancer cell lines by Sulforhodamine B assay.

Files

bib-4efe55da-df74-44d0-860c-14e5d88bb616.txt

Files (346 Bytes)

Name Size Download all
md5:abf8c3cd12a09b0d000a4a654c2e3d4f
346 Bytes Preview Download